[HSF] Aprotinin

Ben Bidstrup benjamin.bidstrup at bigpond.com
Mon Nov 20 13:25:37 EST 2006


http://www.fda.gov/ohrms/dockets/ac/cder06.html#CardiovascularRenal

>  > do you have a link?
>
>NFA
>
>>  -----Original Message-----
>>  From: openheart-l-bounces at lists.hsforum.com [mailto:openheart-l-
>>  bounces at lists.hsforum.com] On Behalf Of Michael Firstenberg
>>  Sent: Sunday, November 19, 2006 7:20 PM
>>  To: OpenHeart-L at lists.hsforum.com
>>  Subject: Re: [HSF] Aprotinin
>>
>>  do you have a link?
>>
>>  michael
>>
>>
>>  On Nov 19, 2006, at 7:16 PM, Ben Bidstrup wrote:
>>
>>  > You might find it interesting to read the FDA transcript of the
>>  > Cardiovascular and Renal Advisory  Board 21 September.
>>  >
>>  >> Please don't disparage Dennis Mangano too much.  He is, or at
>>  >> least was, a
>>  >> very capable clinical cardiac anesthesiologist and is fully
>>  >> cognizant of all
>>  >> of the issues regarding intra-operative bleeding and post-
>>  >> operative care of
>>  >> cardiac surgery patients.  That explains Dennis' consistent
>>  >> ability to focus
>>  >> and publish provocatively on real life issues that confronting
>>  >> surgeons and
>>  >> anesthesiologists on a day to day basis.  The methodology of his
>>  >> paper in
>>  >> the NEJM is open to question.  Dr. Mangano's credentials are not!
>>  >> Fraser Keith
>>  >>
>>  >> -----Original Message-----
>>  >> From: openheart-l-bounces at lists.hsforum.com
>>  >> [mailto:openheart-l-bounces at lists.hsforum.com] On Behalf Of Michael
>>  >> Firstenberg
>>  >> Sent: Sunday, November 19, 2006 10:18 AM
>>  >> To: OpenHeart-L at lists.hsforum.com
>>  >> Subject: Re: [HSF] Aprotinin
>>  >>
>>  >> If I recall Mangino is not a surgeon - in fact is he not an
>>  >> anesthesiologist, as are many of the people who recently write
>>  >> these articles about "bad cardiac drugs"?  Has he actually had to
>>  >> stand at the foot of a bed or in the OR for countless hours
>>  >> watching patient bleed to death and deal first hand with the
>>  >> consequences of massive transfusions.  Yes, renal failure and
>>  >> dialysis is bad bad bad - but compare that with right heart
>>  >> failure/ARDS/massive pressor requirements/etc from excessive
>>  >> bleeding (and the hypotension and associated ATN/renal failure
>>  >> anyhow).  My guess is he is home in bed all nice an cozy with his
>>  >> pager off at the end of his shift.
>>  >>
>>  >> -michael
>>  >>
>>  >>
>>  >>
>>  >>
>>  >> On Nov 19, 2006, at 2:24 AM, Ani Anyanwu wrote:
>>  >>
>>  >>>  Prasanna
>>  >>>
>>  >>>  Well many would I suspect call it unbridled.
>>  >>>
>>  >>>  The following would generally receive aprotinin in my institution
>>  >>>  1) reoperations
>>  >>>  2) operations on the aortic arch or descending aorta
>>  >>>  3) transplant and VAD procedures
>>  >>>  4) operations on patients on clopidogrel
>>  >>>  5) combined valvular and CABG
>>  >>>  6) Patients with renal impairment
>>  >>>  7) Patients where ability to tolerate transfusion or bleeding
>>  >>> complications is thought to be marginal including - most
>>  >>> patients  aged 70 or above, patients with severe lung disease,
>>  >>> poor LV  function, severe pulmonary hypertension, multiple
>>  >>> comorbidity etc.  Certainly almost all octogenrians would get
>>  >>> aprotinin - even for CABG.
>  > >>>  8) Paradoxically, young patients in their 20s or 30s (where
>>  >>> avoidance of blood transfusion should be the goal in all patients)
>>  >>>  9) Multiple valvular procedures (excluding tricuspid valve)
>>  >>>  10) cases with anticipated bypass run more than 3 hours
>>  >>> (including  complex mitral repairs)
>>  >>>
>>  >>>  As you can see there is not much left - so maybe it is
>>  >>> unbridled!  As you implied we obviously would not use it for an
>>  >>> ASD or isolated  AVR, but these constitute a small minority of
>>  >>> our procedures.  Personally I would use it for practically every
>>  >>> operation -  including all CABGs - but that is a personal opinion
>>  >>> as I believe  there are non-hematological benefits of the drug
>>  >>> and like you
>>  >>  > strongly believe in blood conservation. I do not have any
>>  >> interests
>>  >>>  or links to industry.
>>  >>>
>>  >>>  Actually Ben brought up something that I had never thought of -
>  > >>> correct me if I am wrong but Aprotinin is the only agent
>>  >>> licensed  as a blood conservation agent for heart surgery?
>>  >>>
>>  >>>  Ani
>>  >>>    ----- Original Message -----
>>  >>>    From: psimha<mailto:prasannasimha at gmail.com>
>>  >>>    To: OpenHeart-L at lists.hsforum.com<mailto:OpenHeart-
>>  >>>  L at lists.hsforum.com>
>>  >>>    Sent: Sunday, November 19, 2006 12:00 AM
>>  >>>    Subject: Re: [HSF] Aprotinin
>>  >>>
>>  >>>
>>  >>>    Ani - are you really using it "unbridled" or liberally ? Do
>>  >>> you  use it
>>  >>>    for an ASD or for a straight forward valve replacement ? or
>>  >>> any  other
>>  >>>    case with a short bypass run ?
>>  >>>    I did not say I will not use it in a redo - in fact if you
>>  >>> note my
>>  >>>    original post I said I did use it in redo's ?
>>  >>>    And Yes , I believe very strongly in blood conservation and
>>  >>> believe that
>>  >>>    Aprotinin is one (and not the only ) cog in the wheel.
>>  >>  >   Prasanna
>>  >>>
>>  >>>    Ani Anyanwu wrote:
>>  >>>>  Prasanna
>>  >>>>
>>  >>>>  We use aprotinin in an unbridled way and are certainly yet to
>>  >>>> see  this price.
>>  >>>>  - we have no more an incidence of renal failure than other
>>  >>>> institutions have (this we know because incidence of dialysis
>>  >>>> postop in all New York Hospitals is tracked by the State
>>  >>>> Department of Health)
>>  >>>>  - we have no suggestion of an increase in early vein graft
>>  >>>> thrombosis (this should transform into higher periop MI and
>>  >>>> mortality, our CABG mortality rate has remained around 1.5% last
>>  >>>> 3  years)
>>  >>>>  - we have not experienced any adverse events that caused us to
>>  >>>> be  concerned about its use, except fatal thrombosis in 2
>>  >>>> patients  with Factor V Lieden deficiency having circulatory
>>  >>>> arrest so we  now routinely screen for this defect in all
>>  >>>> circulatory arrest cases.
>>  >>>>
>>  >>>>  The price we are paying is a low incidence of transfusion of
>>  >>>> blood  products and a low re-exploration rate (<2% last 2 years
>>  >>>> even with  18% being redos and almost 20% aortic cases). Maybe
>>  >>>> there are  other unknown adverse effects which will catch up
>>  >>>> with us, but for  know they are unknown (and we wont be
>>  >>>> responsible; remember it is  the drug companies not doctors
>>  >>>> being sued for COX2 inhibitors).
>>  >>>>
>>  >>>>  Maybe when Mangano is bored he might do another study, and
>>  >>>> then  what will you do? For those who use Amicar, how do we
>>  >>>> really know  it is any safer - the drug is not even licensed for
>>  >>>> human use in  many European countries. Perhaps even his next
>>  >>>> study will be on  morbidity of plasma and platelet
>>  >>>> transfusions....then what will we  do?
>>  >>>>
>>  >>>>  Ani
>>  >>>>    ----- Original Message -----
>>  >>>>    From:
>>  >>>> prasannasimha<mailto:prasannasimha at gmail.com<mailto:prasannasimha at g
>>  >>>> ma
>>  >>>>  il.com>>
>>  >>>>    To: OpenHeart-L at lists.hsforum.com<mailto:OpenHeart-
>>  >>>>  L at lists.hsforum.com<mailto:OpenHeart-
>>  >>>>  L at lists.hsforum.com<mailto:OpenHeart-L at lists.hsforum.com>>
>>  >>>>    Sent: Saturday, November 18, 2006 9:37 PM
>>  >>>>    Subject: Re: [HSF] Aprotinin
>>  >>>>
>>  >>>>
>>  >>>>    The thing I want to say is that be it Vioxx / Aprotinin/blood/
>  > >>>>  Oxygen -
>>  >>>>    they are all drugs and have effects and side effects. The
>>  >>>> present mess
>>  >>>>    that the pharmacological companies are in is just because of
>>  >>>> their
>>  >>>>    unbridled enthusiasm (or greed) to ,make a quick buck and it
>>  >>>> backfires
>>  >>>>    on them. COX2 Inhibitors have a specific role unfortunately
>>  >>>> I  even saw
>>  >>>>    my dentist prescribing it for tooth pain !! Who marketed it
>>  >>>> to  him as a
>>  >>>>    good NSAID  ? I told him about the literature and my
>>  >>>> concerns  (this was
>>  >>>>    prior to Vioxx) . They were trying to market Valdecoxib for
>>  >>>> post  cardiac
>>  >>>>    surgery pain !!_ and I told them you should not be doing that
>>  >>>> -  but did
>>  >>>>    they listen ? and bang in a few months a controversy breaks
>>  >>>> out.  The
>>  >>>>    wife of colleague of mine was taking valdecoxib sample (she
>  > >>>> is a  Doctor
>>  >>>>    too) as the sample was around and the premenopausal lady
>>  >>>> ended  up with a
>>  >>>>    coronary thrombosis !!
>>  >>>>    Every drug has a role and an indication based on good
>>  >>>> clinical  judgment
>>  >>  >>   - unfortunately we pay the price when its use is unbridled.
>>  >>>>    Prasanna
>>  >>>>
>>  >>>>
>>  hgrmd at aol.com<mailto:hgrmd at aol.com<mailto:hgrmd at aol.com<mailto:hgrm
>>  >>>> d@
>>  >>>>  aol.com>> wrote:
>>  >>>>>  Prasanna and Ajit,
>>  >>>>>    At the risk of great bodily harm from Ben, Ani, and others,
>>  >>>>> I  again think the use of aprotinin should be limited as much
>>  >>>>> as  possible.  I know there are cases where the benefit
>>  >>>>> seemingly  outweighs the risk.  However, the mounting
>>  >>>>> literature against it  is becoming increasingly compelling.  In
>>  >>>>> addition, my own  impression, made years before any of this
>>  >>>>> came out, was that the  drug increased the risk of ATN.  I'm
>>  >>>>> also convinced that this has  the potential to be the Vioxx of
>>  >>>>> cardiac surgery.  All I can say  is you guys who continue to
>>  >>>>> indiscriminantly use it have got some  really big ones.
>>  >>>>>  Hal
>>  >>>>>
>>  >>>>>
>>  >>>>>  -----Original Message-----
>>  >>>>>  From:
>>  >>>>> prasannasimha at gmail.com<mailto:prasannasimha at gmail.com<mailto:pras
>>  >>>>> an
>>  >>>>>  nasimha at gmail.com<mailto:prasannasimha at gmail.com>>
>>  >>>>>  To: OpenHeart-L at lists.hsforum.com<mailto:OpenHeart-
>>  >>  >>> L at lists.hsforum.com<mailto:OpenHeart-
>>  >>>>>  L at lists.hsforum.com<mailto:OpenHeart-L at lists.hsforum.com>>
>>  >>>>>  Sent: Sat, 18 Nov 2006 1:00 PM
>>  >>>>>  Subject: Re: [HSF] Aprotinin
>>  >>>>>
>>  >>>>>
>>  >>>>>  Very Sorry used Aprotinin on my redo - can't help using it
>>  >>>>> selectively !!
>>  >>>>>  Prasanna
>>  >>>>>
>>  >>>>>  Ajit Damle wrote:
>>  >>>>>
>>  >>>>>>  Journal club critique >
>>  >>>>>>  A disheartening story: Aprotinin in cardiac surgery >
>>  >>>>>>  Lien M, Milbrandt E
>>  >>>>>>
>>  >>>>>>  Critical Care, 2006 10:317 ( 8 November 2006 )
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  Journal club critique
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  A disheartening story: Aprotinin in cardiac surgery
>>  >>>>>>
>>  >>>>>>  Marcus Lien1 and Eric B Milbrandt2 >
>>  >>>>>>  1Clinical Fellow, Department of Critical Care Medicine,
>>  >>>>>> University of
>>  >>>>>>  Pittsburgh School of Medicine, Pittsburgh, Pennsylvania, USA
>>  >>>>>>
>>  >>>>>>  2Assistant Professor, Department of Critical Care Medicine,
>>  >>>>>> University of
>>  >>>>>>  Pittsburgh School of Medicine, Pittsburgh, Pennsylvania, USA
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  Critical Care 2006, 10:317 doi:10.1186/cc5072
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>>
>>  >>>>>>>
>>  >>>>>>  Evidence based medicine journal club critique edited by E B
>>  >>>>>> Milbrant
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  The electronic version of this article is the complete one
>>  >>>>>> and  can be found
>>  >>>>>>  online at: http://ccforum.com/content/10/6/317<http://
>>  >>>>>>  ccforum.com/content/10/6/317<http://ccforum.com/content/
>>  >>>>>>  10/6/317<http://ccforum.com/content/10/6/317>>
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  Published 8 November 2006 >
>>  >>>>>>
>>  >>>>>>  C 2006 BioMed Central Ltd
>>  >>>>>>
>>  >>>>>>  Citation
>>  >>>>>>
>>  >>>>>>  Mangano DT, Tudor IC, Dietzel C: The risk associated with
>  > >>>>>> aprotinin in
>>  >>>>>>  cardiac surgery. N Engl J Med 2006, 354:353-365 [1].
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  Background
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  The majority of patients undergoing surgical treatment for ST-
>>  >>>>>>  elevation
>>  >>>>>>  myocardial infarction receive antifibrinolytic therapy to
>>  >>>>>> limit  blood loss.
>>  >>>>>>  This approach appears counterintuitive to the accepted
>>  >>>>>> medical  treatment of
>>  >>>>>>  the same condition - namely, fibrinolysis to limit
>>  >>>>>> thrombosis.  Despite this
>>  >>>>>>  concern, no independent, large-scale safety assessment has
>>  >>>>>> been  undertaken.
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  Methods
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  Design and setting
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  Prospective observational cohort study in 69 institutions in
>>  >>>>>> North and South
>>  >>>>>>  America, the Middle East, Europe, and Asia.
>>  >>>>>>
>  > >>>>>>
>>  >>>>>>  Subjects
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  4374 patients undergoing coronary-artery revascularization.
>>  >>>>>> All  patients
>>  >>>>>>  were >18 years old and completed a pre-surgery interview.
>>  >>>>>> Patients were
>>  >>>>>>  classified as undergoing primary surgery (no previous heart
>>  >>>>>> surgery and no
>>  >>>>>>  other surgery besides a coronary artery bypass graft), or
>>  >>>>>> complex surgery
>>  >>>>>>  (all other surgery).
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  Intervention
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  None.
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  Measurements
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  The authors prospectively assessed three agents (aprotinin
>>  >>>>>> [1295  patients],
>>  >>>>>>  aminocaproic acid [883], and tranexamic acid [822]) as
>>  >>>>>> compared  with no
>>  >>>>>>  agent (1374 patients) with regard to serious cardiovascular,
>>  >>  >>>> renal, and
>>  >>>>>>  cerebrovascular outcomes by propensity and multivariable
>>  >>>>>> methods.
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  Results
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  In propensity-adjusted, multivariable logistic regression (C-
>>  >>>>>>  index, 0.72),
>>  >>>>>>  use of aprotinin was associated with a doubling in the risk
>>  >>>>>> of  renal failure
>>  >>>>>>  requiring dialysis among patients undergoing complex coronary-
>>  >>>>>>  artery surgery
>>  >>>>>>  (odds ratio, 2.59; 95 percent confidence interval, 1.36 to
>>  >>>>>> 4.95)  or primary
>>  >>>>>>  surgery (odds ratio, 2.34; 95 percent confidence interval,
>>  >>>>>> 1.27  to 4.31).
>>  >>>>>>  Similarly, use of aprotinin in the latter group was
>>  >>>>>> associated  with a 55
>>  >>>>>>  percent increase in the risk of myocardial infarction or
>>  >>>>>> heart  failure (P <
>>  >>>>>>  0.001) and a 181 percent increase in the risk of stroke or
>>  >>>>>> encephalopathy (P
>>  >>>>>>  = 0.001). Neither aminocaproic acid nor tranexamic acid was
>>  >>>>>> associated with
>>  >>>>>>  an increased risk of renal, cardiac, or cerebral events.
>>  >>>>>> Adjustment
>>  >>>>>>  according to propensity score for the use of any one of the
>>  >>>>>> three agents as
>>  >>>>>>  compared with no agent yielded nearly identical findings. All
>>  >>  >>>> the agents
>>  >>>>>>  reduced blood loss.
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  Conclusion
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  The association between aprotinin and serious end-organ
>>  >>>>>> damage  indicates
>>  >>>>>>  that continued use is not prudent. In contrast, the less
>>  >>>>>> expensive generic
>>  >>>>>>  medications aminocaproic acid and tranexamic acid are safe
>>  >>>>>> alternatives.
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>>
>>  >>>>>>  The medical and surgical approaches to acute ST-elevation
>>  >>>>>> myocardial
>>  >>>>>>  infarction present an interesting paradox. The medical
>>  >>>>>> approach  focuses on
>>  >>>>>>  fibrinolytic therapy. Due to concerns over bleeding, the
>>  >>>>>> surgical approach
>>  >>>>>>  avoids fibrinolytic agents and instead uses agents that
>>  >>>>>> mitigate  bleeding,
>>  >>>>>>  so called antifibrinolytic agents, which include aprotinin,
>>  >>>>>> aminocaproic
>>  >>>>>>  acid, and tranexamic acid. These agents were generally
>>  >>>>>> considered safe based
>>  >>>>>>  on a number of secondary analyses of studies that were not
>>  >>>>>> primarily
>>  >>>>>>  intended to assess safety. These relatively small studies
>  > >>>>>> were  underpowered
>>  >>>>>>  to detect adverse events and did not involve head-to-head
>>  >>>>>> comparisons of the
>>  >>>>>>  commonly used antifibrinolytic agents. Animal studies
>>  >>>>>> suggest  that these
>>  >>>>>>  agents have the potential to cause ischemic damage to
>>  >>>>>> multiple  organ systems
>>  >>>>>>  and small, largely single-center studies have suggested
>>  >>>>>> increased graft
>>  >>>>>>  thrombosis and renal dysfunction [2-6]. Ideally, the safety
>>  >>>>>> of  these agents
>>  >>>>>>  would be compared in a large, multi-center, randomized
>>  >>>>>> controlled trial.
>>  >>>>>>  However, because their use is embedded in practice and
>>  >>>>>> because  regulatory
>>  >>>>>>  approval of these agents differs by country, conducting such
>>  >>>>>> a  trial will be
>>  >>>>>>  difficult if not impossible.
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  To address the safety of these agents for cardiopulmonary
>  > >>>>>> bypass  surgery,
>>  >>>>>>  Mangano and colleagues [1] conducted a large, prospective,
>>  >>>>>> observational
>>  >>>>>>  cohort assessing aprotinin, aminocaproic acid, and
>>  >>>>>> tranexamic  acid as
>>  >>>>>>  compared to no agent in 4374 patients undergoing
>>  >>>>>> revascularization. Because
>>  >>>>>>  this was a prospective study, the authors were able to
>>  >>>>>> collect a  wealth of
>>  >>>>>>  clinical information, including approximately 7500 data
>>  >>>>>> fields  per patient.
>>  >>>>>>  This permitted consideration of variables that might
>>  >>>>>> influence  both choice
>>  >>>>>>  of antifibrinolytic agent and clinical outcome. The authors
>>  >>>>>> used a
>>  >>>>>>  propensity score based on 45 treatment-selection covariates and
>>  >>>>>>  multivariable modeling to control for baseline differences
>>  >>>>>> between groups.
>>  >>>>>>  In doing so, they found that aprotinin, but not aminocaproic
>>  >>>>>> acid or
>>  >>>>>>  tranexamic acid, was associated with serious cardiovascular,
>>  >>>>>> renal, and
>>  >>>>>>  cerebrovascular adverse events. Furthermore, a dose-response
>>  >>>>>> relationship
>>  >>>>>>  was demonstrated, strengthening the inference of causality.
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  The main weakness of this study is that the authors failed to
>>  >>  >>>> report details
>>  >>>>>>  of the surgery itself, such as whether the surgery was on
>>  >>>>>> vs.  off-pump, time
>>  >>>>>>  on pump, and number of vessels bypassed. These variables are
>>  >>>>>> likely to
>>  >>>>>>  influence not only choice of antifibrinolytic agent but also
>>  >>>>>> outcome, and
>>  >>>>>>  are, therefore, a source of indication bias that could
>>  >>>>>> reflect  unfavorably
>>  >>>>>>  on aprotinin.
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  Based on the results of this study and those of another
>>  >>>>>> observational study
>>  >>>>>>  suggesting renal toxicity [7], the United States Food and Drug
>>  >>>>>>  Administration (FDA) held an advisory committee meeting
>>  >>>>>> September 21, 2006
>>  >>>>>>  to consider the cardiovascular safety of aprotinin. Because
>>  >>>>>> of  concerns
>>  >>>>>>  about the methodology of the study by Mangano and colleagues
>>  >>>>>> and  because it
>>  >>>>>>  was the only study to suggest cardiovascular adverse events
>>  >>>>>> [8],  the
>>  >>>>>>  advisory committee concluded that there was insufficient
>>  >>>>>> evidence to support
>>  >>>>>>  changing the cardiovascular safety labeling of the drug.
>>  >>>>>> However, just six
>>  >>>>>>  days after the committee met, it was revealed that the
>>  >>>>>> drug's  manufacturer,
>>  >>  >>>> Bayer, had preliminary results from an observational study of
>>  >>>>>>  67,000 cardiac
>>  >>>>>>  bypass patients that suggested aprotinin was associated with
>>  >>>>>> increased risk
>>  >>>>>>  of death, renal dysfunction, congestive heart failure, and
>>  >>>>>> stroke [9]. The
>>  >>>>>>  FDA subsequently issued a statement indicating it was unaware
>>  >>>>>> of  this study
>>  >>>>>>  when the advisory committee met and that it is evaluating
>>  >>>>>> the  results of
>>  >>>>>>  this study and the potential implications for the use of
>>  >>>>>> aprotinin [10]. In
>>  >>>>>>  the mean time, the FDA suggests that physicians who use
>>  >>>>>> aprotinin should
>  > >>>>>>  carefully monitor patients for the occurrence of toxicity,
>>  >>>>>> particularly to
>>  >>>>>>  the kidneys, heart, or brain, and promptly report observed
>>  >>>>>> adverse events.
>>  >>>>>>  They go on to recommend that physicians should consider
>>  >>>>>> limiting  aprotinin
>>  >>>>>>  use to those situations where the clinical benefit of
>>  >>>>>> reduced  blood loss is
>>  >>>>>>  essential to medical management of the patient and outweighs
>>  >>>>>> the  potential
>>  >>>>>>  risks.
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  Recommendation >
>>  >>>>>>
>>  >>>>>>  The weight of evidence suggests that aprotinin increases the
>>  >>>>>> risk for a poor
>>  >>>>>>  outcome among patients undergoing cardiac operations. Not
>>  >>>>>> only  is this drug
>>  >>>>>>  very expensive, it seems to be toxic. Although the risk of
>>  >>>>>> excessive
>>  >>>>>>  bleeding is certainly a cause for concern in certain
>>  >>>>>> patients,  and treatment
>  > >>>>>>  with aprotinin can decrease blood loss in selected patients,
>>  >>>>>> data are
>>  >>>>>>  lacking to show that administration of this agent actually
>>  >>>>>> improves
>>  >>>>>>  survival.
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  Competing interests
>>  >>>>>>
>>  >>>>>>  The authors declare that they have no competing interests.
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>>
>>  >>>>>>  1. Mangano DT, Tudor IC, Dietzel C: The risk associated with
>>  >>>>>> aprotinin in
>>  >>>>>>  cardiac surgery.
>>  >>>>>>
>>  >>>>>>  N Engl J Med 2006, 354:353-365. >
>>  >>>>>>
>>  >>>>>>  2. Cosgrove DM III, Heric B, Lytle BW, Taylor PC, Novoa R,
>>  >>>>>> Golding LA,
>>  >>>>>>  Stewart RW, McCarthy PM, Loop FD: Aprotinin therapy for
>>  >>>>>> reoperative
>>  >>>>>>  myocardial revascularization: a placebo-controlled study.
>>  >>>>>>
>>  >>>>>>  Ann Thorac Surg 1992, 54:1031-1036.
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  3. D'Ambra MN, Akins CW, Blackstone EH, Bonney SL, Cohn LH,
>>  >>>>>> Cosgrove DM,
>>  >>>>>>  Levy JH, Lynch KE, Maddi R: Aprotinin in primary valve
>>  >>>>>> replacement and
>>  >>>>>>  reconstruction: a multicenter, double-blind, placebo-
>>  >>>>>> controlled  trial.
>>  >>>>>>
>>  >>>>>>  J Thorac Cardiovasc Surg 1996, 112:1081-1089
>>  >>>>>>
>>  >>>>>>
>>  >>>>>>  4. Feindt PR, Walcher S, Volkmer I, Keller HE, Straub U,
>>  >>>>>> Huwer  H, Seyfert
>>  >>>>>>  UT, Petzold T, Gams E: Effects of high-dose aprotinin on
>>  >>>>>> renal  function in
>>  >>>>>>  aortocoronary bypass grafting.
>>  >>>>>>
>>  >>>>>>  Ann Thorac Surg 1995, 60:1076-1080 >
>>  >>>>>>
>>  >>>>>>  5. Sundt TM III, Kouchoukos NT, Saffitz JE, Murphy SF,
>>  >>>>>> Wareing  TH, Stahl
>>  >>>>>>  DJ: Renal dysfunction and intravascular coagulation with
>>  >>>>>> aprotinin and
>>  >>>>>>  hypothermic circulatory arrest.
>>  >>  >>>>
>>  >>>>>>  Ann Thorac Surg 1993, 55:1418-1424 >
>>  >>>>>>
>>  >>>>>>  6. Umbrain V, Christiaens F, Camu F: Intraoperative coronary
>>  >>>>>> thrombosis:
>>  >>>>>>  can aprotinin and protamine be incriminated?
>>  >>>>>>
>>  >>>>>>  J Cardiothorac Vasc Anesth 1994, 8:198-201 >
>>  >>>>>>
>>  >>>>>>  7. Karkouti K, Beattie WS, Dattilo KM, McCluskey SA, Ghannam
>>  >>>>>> M,  Hamdy A,
>>  >>>>>>  Wijeysundera DN, Fedorko L, Yau TM: A propensity score case-
>>  >>>>>> control
>>  >>>>>>  comparison of aprotinin and tranexamic acid in high-transfusion-
>>  >>>>>>  risk cardiac
>>  >>>>>>  surgery.
>>  >>>>>>
>>  >>>>>>  Transfusion 2006, 46:327-338 >
>>  >>>>>>
>>  >>>>>>  8. Hughes S: Aprotinin safety again in spotlight as new
>>  >>>>>> study  suggests
>>  >>>>>>  increased cardiac events.
>>  >>>>>>
>>  >>>>>>  http://www.medscape.com/viewarticle/545400<http://
>>  >>>>>>  www.medscape.com/viewarticle/545400<http://www.medscape.com/
>>  >>>>>>  viewarticle/545400<http://www.medscape.com/viewarticle/
>>  >>>>>> 545400>> >
>>  >>>>>>  October 2, 2006 >
>>  >>>>>>  9. Harris G: FDA says Bayer failed to reveal drug risk study.
>>  >>>>>>
>>  >>>>>>  [http://www.nytimes.com/2006/09/30/health/30fda.html] New
>>  >>>>>> York  Times >
>>  >>>>>>
>>  >>>>>>  10. US Food and Drug Administration: FDA Public Health
>>  >>>>>> Advisory:  Aprotinin
>>  >>>>>>  Injection (marketed as Trasylol).
>>  >>>>>>
>>  >>>>>>  [http://www.fda.gov/cder/drug/advisory/aprotinin20060929.htm] >
>>  >>  >>>> September 29, 2006 >
>  > >>>>>>
>>  >>>>>>  _______________________________________________
>>  >>>>>>  OpenHeart-L mailing list
>>  >>>>>>
>>  >>>>>>  Send postings to:
>>  >>>>>>  OpenHeart-L at lists.hsforum.com<mailto:OpenHeart-
>>  >>>>>>  L at lists.hsforum.com<mailto:OpenHeart-
>>  >>>>>>  L at lists.hsforum.com<mailto:OpenHeart-L at lists.hsforum.com>>
>>  >>>>>>
>>  >>>>>>  To UNSUBSCRIBE, to CHANGE email address, or to view archives:
>>  >>>>>>  http://mmp.cjp.com/mailman/listinfo/openheart-l<http://
>>  >>>>>>  mmp.cjp.com/mailman/listinfo/openheart-l<http://mmp.cjp.com/
>>  >>>>>>  mailman/listinfo/openheart-l<http://mmp.cjp.com/mailman/
>>  >>>>>> listinfo/
>>  >>>>>>  openheart-l>>
>>  >>>>>>
>>  >>>>>>  All messages transmitted by the OpenHeart-L are subject to
>>  >>>>>> the  policies and > disclaimers posted at:
>>  >>>>>>  http://www.hsforum.com/listdisclaim<http://www.hsforum.com/
>>  >>>>>>  listdisclaim<http://www.hsforum.com/listdisclaim<http://
>>  >>>>>>  www.hsforum.com/listdisclaim>>
>  > >>>>>>  -----------------------------------------
>>  >>>>>>
>>  >>>>>>  _______________________________________________
>>  >>>>>>
>>  >>>>>  OpenHeart-L mailing list
>>  >>>>>
>>  >>>>>  Send postings to:
>>  >>>>>  OpenHeart-L at lists.hsforum.com<mailto:OpenHeart-
>>  >>>>>  L at lists.hsforum.com<mailto:OpenHeart-
>>  >>>>>  L at lists.hsforum.com<mailto:OpenHeart-L at lists.hsforum.com>>
>>  >>>>>
>>  >>>>>  To UNSUBSCRIBE, to CHANGE email address, or to view archives:
>>  >>>>>  http://mmp.cjp.com/mailman/listinfo/openheart-l<http://
>>  >>>>>  mmp.cjp.com/mailman/listinfo/openheart-l<http://mmp.cjp.com/
>>  >>>>>  mailman/listinfo/openheart-l<http://mmp.cjp.com/mailman/listinfo/
>>  >>>>>  openheart-l>>
>>  >>>>>
>>  >>>>>  All messages transmitted by the OpenHeart-L are subject to
>>  >>>>> the  policies and disclaimers posted at:
>>  >>>>>  http://www.hsforum.com/listdisclaim<http://www.hsforum.com/
>>  >>>>>  listdisclaim<http://www.hsforum.com/listdisclaim<http://
>>  >>>>>  www.hsforum.com/listdisclaim>>
>>  >>>>>  -----------------------------------------
>>  >>>>>
>>  >>>>>
>>  __________________________________________________________________
>>  >>>>> __
>>  >>>>>  ____
>>  >>>>>  Check out the new AOL.  Most comprehensive set of free safety
>>  >>>>> and  security tools, free access to millions of high-quality
>>  >>>>> videos  from across the web, free AOL Mail and more.
>>  >>>>>  _______________________________________________
>>  >>>>>  OpenHeart-L mailing list
>>  >>>>>
>>  >>>>>  Send postings to:
>>  >>>>>   OpenHeart-L at lists.hsforum.com<mailto:OpenHeart-
>>  >>>>>  L at lists.hsforum.com<mailto:OpenHeart-
>>  >>>>>  L at lists.hsforum.com<mailto:OpenHeart-L at lists.hsforum.com>>
>>  >>>>>
>>  >>>>>  To UNSUBSCRIBE, to CHANGE email address, or to view archives:
>>  >>>>>  http://mmp.cjp.com/mailman/listinfo/openheart-l<http://
>>  >>>>>  mmp.cjp.com/mailman/listinfo/openheart-l<http://mmp.cjp.com/
>>  >>>>>  mailman/listinfo/openheart-l<http://mmp.cjp.com/mailman/listinfo/
>>  >>>>>  openheart-l>>
>>  >>>>>
>>  >>>>>  All messages transmitted by the OpenHeart-L are subject to
>>  >>>>> the  policies and
>>  >>>>>  disclaimers posted at:
>>  >>>>>  http://www.hsforum.com/listdisclaim<http://www.hsforum.com/
>>  >>>>>  listdisclaim<http://www.hsforum.com/listdisclaim<http://
>>  >>  >>> www.hsforum.com/listdisclaim>>
>>  >>>>>  -----------------------------------------
>>  >>>>>
>>  >>>>>
>>  >>>>>
>>  >>>>
>>  >>>>    _______________________________________________
>>  >>>>    OpenHeart-L mailing list
>>  >>>>
>>  >>>>    Send postings to:
>>  >>>>     OpenHeart-L at lists.hsforum.com<mailto:OpenHeart-
>>  >>>>  L at lists.hsforum.com<mailto:OpenHeart-
>>  >>>>  L at lists.hsforum.com<mailto:OpenHeart-L at lists.hsforum.com>>
>>  >>>>
>>  >>>>    To UNSUBSCRIBE, to CHANGE email address, or to view archives:
>>  >>>>    http://mmp.cjp.com/mailman/listinfo/openheart-l<http://
>>  >>>>  mmp.cjp.com/mailman/listinfo/openheart-l<http://mmp.cjp.com/
>>  >>>>  mailman/listinfo/openheart-l<http://mmp.cjp.com/mailman/listinfo/
>>  >>>>  openheart-l>>
>>  >>>>
>>  >>>>    All messages transmitted by the OpenHeart-L are subject to
>>  >>>> the  policies and
>>  >>>>    disclaimers posted at:
>>  >>>>    http://www.hsforum.com/listdisclaim<http://www.hsforum.com/
>  > >>>>  listdisclaim<http://www.hsforum.com/listdisclaim<http://
>>  >>>>  www.hsforum.com/listdisclaim>>
>>  >>>>    -----------------------------------------
>>  >>>>  _______________________________________________
>>  >>>>  OpenHeart-L mailing list
>>  >>>>
>>  >>>>  Send postings to:
>>  >>>>   OpenHeart-L at lists.hsforum.com<mailto:OpenHeart-
>>  >>>> L at lists.hsforum.com>
>>  >>>>
>>  >>>>  To UNSUBSCRIBE, to CHANGE email address, or to view archives:
>>  >>>>  http://mmp.cjp.com/mailman/listinfo/openheart-l<http://
>>  >>>> mmp.cjp.com/
>>  >>  >> mailman/listinfo/openheart-l>
>>  >>>>
>>  >>>>  All messages transmitted by the OpenHeart-L are subject to the
>>  >>>> policies and
>>  >>>>  disclaimers posted at:
>>  >>>>  http://www.hsforum.com/listdisclaim<http://www.hsforum.com/
>>  >>>>  listdisclaim>
>>  >>>>  -----------------------------------------
>>  >>>>
>>  >>>>
>>  >>>>
>>  >>>
>>  >>>    _______________________________________________
>>  >>>    OpenHeart-L mailing list
>  > >>>
>>  >>>    Send postings to:
>>  >>>     OpenHeart-L at lists.hsforum.com<mailto:OpenHeart-
>>  >>> L at lists.hsforum.com>
>>  >>>
>>  >>>    To UNSUBSCRIBE, to CHANGE email address, or to view archives:
>>  >>>    http://mmp.cjp.com/mailman/listinfo/openheart-l<http://
>>  >>>  mmp.cjp.com/mailman/listinfo/openheart-l>
>>  >>>
>>  >>>    All messages transmitted by the OpenHeart-L are subject to
>>  >>> the  policies and
>>  >>>    disclaimers posted at:
>>  >>>    http://www.hsforum.com/listdisclaim<http://www.hsforum.com/
>>  >>>  listdisclaim>
>>  >>>    -----------------------------------------
>>  >>>  _______________________________________________
>>  >>>  OpenHeart-L mailing list
>>  >>>
>>  >>>  Send postings to:
>>  >>>   OpenHeart-L at lists.hsforum.com
>>  >>>
>>  >>>  To UNSUBSCRIBE, to CHANGE email address, or to view archives:
>>  >>>  http://mmp.cjp.com/mailman/listinfo/openheart-l
>>  >>>
>>  >>>  All messages transmitted by the OpenHeart-L are subject to the
>>  >>> policies and
>>  >>>  disclaimers posted at:
>>  >>>  http://www.hsforum.com/listdisclaim
>>  >>>  -----------------------------------------
>>  >>
>>  >> _______________________________________________
>>  >> OpenHeart-L mailing list
>>  >>
>>  >> Send postings to:
>>  >>  OpenHeart-L at lists.hsforum.com
>>  >>
>>  >> To UNSUBSCRIBE, to CHANGE email address, or to view archives:
>>  >> http://mmp.cjp.com/mailman/listinfo/openheart-l
>>  >>
>>  >> All messages transmitted by the OpenHeart-L are subject to the
>>  >> policies and
>>  >> disclaimers posted at:
>>  >> http://www.hsforum.com/listdisclaim
>>  >> -----------------------------------------
>>  >>
>>  >> _______________________________________________
>>  >> OpenHeart-L mailing list
>>  >>
>>  >> Send postings to:
>>  >>  OpenHeart-L at lists.hsforum.com
>>  >>
>>  >> To UNSUBSCRIBE, to CHANGE email address, or to view archives:
>>  >> http://mmp.cjp.com/mailman/listinfo/openheart-l
>>  >>
>>  >> All messages transmitted by the OpenHeart-L are subject to the
>>  >> policies and
>>  >> disclaimers posted at:
>>  >> http://www.hsforum.com/listdisclaim
>>  >> -----------------------------------------
>>  >
>>  >
>>  > --
>>  > Ben Bidstrup FRACS FRCSEd FEBCTS
>>  > Consultant Cardiothoracic Surgeon
>>  > _______________________________________________
>>  > OpenHeart-L mailing list
>>  >
>>  > Send postings to:
>>  > OpenHeart-L at lists.hsforum.com
>>  >
>>  > To UNSUBSCRIBE, to CHANGE email address, or to view archives:
>>  > http://mmp.cjp.com/mailman/listinfo/openheart-l
>>  >
>>  > All messages transmitted by the OpenHeart-L are subject to the
>>  > policies and disclaimers posted at:
>>  > http://www.hsforum.com/listdisclaim
>>  > -----------------------------------------
>>
>>  _______________________________________________
>>  OpenHeart-L mailing list
>>
>>  Send postings to:
>>   OpenHeart-L at lists.hsforum.com
>>
>>  To UNSUBSCRIBE, to CHANGE email address, or to view archives:
>>  http://mmp.cjp.com/mailman/listinfo/openheart-l
>>
>>  All messages transmitted by the OpenHeart-L are subject to the policies
>and
>>  disclaimers posted at:
>>  http://www.hsforum.com/listdisclaim
>>  -----------------------------------------
>
>_______________________________________________
>OpenHeart-L mailing list
>
>Send postings to:
>  OpenHeart-L at lists.hsforum.com
>
>To UNSUBSCRIBE, to CHANGE email address, or to view archives:
>http://mmp.cjp.com/mailman/listinfo/openheart-l
>
>All messages transmitted by the OpenHeart-L are subject to the policies and
>disclaimers posted at:
>http://www.hsforum.com/listdisclaim
>-----------------------------------------


-- 
Ben Bidstrup FRACS FRCSEd FEBCTS
Consultant Cardiothoracic Surgeon


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