[HSF] Aprotinin

Nasser F. Abou'Seada nfaabouseada at gmail.com
Mon Nov 20 03:19:54 EST 2006


Thanks Ben .... that has been very helpful ...

NFA

> -----Original Message-----
> From: openheart-l-bounces at lists.hsforum.com [mailto:openheart-l-
> bounces at lists.hsforum.com] On Behalf Of Ben Bidstrup
> Sent: Sunday, November 19, 2006 9:26 PM
> To: OpenHeart-L at lists.hsforum.com
> Subject: RE: [HSF] Aprotinin
> 
> http://www.fda.gov/ohrms/dockets/ac/cder06.html#CardiovascularRenal
> 
> >  > do you have a link?
> >
> >NFA
> >
> >>  -----Original Message-----
> >>  From: openheart-l-bounces at lists.hsforum.com [mailto:openheart-l-
> >>  bounces at lists.hsforum.com] On Behalf Of Michael Firstenberg
> >>  Sent: Sunday, November 19, 2006 7:20 PM
> >>  To: OpenHeart-L at lists.hsforum.com
> >>  Subject: Re: [HSF] Aprotinin
> >>
> >>  do you have a link?
> >>
> >>  michael
> >>
> >>
> >>  On Nov 19, 2006, at 7:16 PM, Ben Bidstrup wrote:
> >>
> >>  > You might find it interesting to read the FDA transcript of the
> >>  > Cardiovascular and Renal Advisory  Board 21 September.
> >>  >
> >>  >> Please don't disparage Dennis Mangano too much.  He is, or at
> >>  >> least was, a
> >>  >> very capable clinical cardiac anesthesiologist and is fully
> >>  >> cognizant of all
> >>  >> of the issues regarding intra-operative bleeding and post-
> >>  >> operative care of
> >>  >> cardiac surgery patients.  That explains Dennis' consistent
> >>  >> ability to focus
> >>  >> and publish provocatively on real life issues that confronting
> >>  >> surgeons and
> >>  >> anesthesiologists on a day to day basis.  The methodology of his
> >>  >> paper in
> >>  >> the NEJM is open to question.  Dr. Mangano's credentials are not!
> >>  >> Fraser Keith
> >>  >>
> >>  >> -----Original Message-----
> >>  >> From: openheart-l-bounces at lists.hsforum.com
> >>  >> [mailto:openheart-l-bounces at lists.hsforum.com] On Behalf Of Michael
> >>  >> Firstenberg
> >>  >> Sent: Sunday, November 19, 2006 10:18 AM
> >>  >> To: OpenHeart-L at lists.hsforum.com
> >>  >> Subject: Re: [HSF] Aprotinin
> >>  >>
> >>  >> If I recall Mangino is not a surgeon - in fact is he not an
> >>  >> anesthesiologist, as are many of the people who recently write
> >>  >> these articles about "bad cardiac drugs"?  Has he actually had to
> >>  >> stand at the foot of a bed or in the OR for countless hours
> >>  >> watching patient bleed to death and deal first hand with the
> >>  >> consequences of massive transfusions.  Yes, renal failure and
> >>  >> dialysis is bad bad bad - but compare that with right heart
> >>  >> failure/ARDS/massive pressor requirements/etc from excessive
> >>  >> bleeding (and the hypotension and associated ATN/renal failure
> >>  >> anyhow).  My guess is he is home in bed all nice an cozy with his
> >>  >> pager off at the end of his shift.
> >>  >>
> >>  >> -michael
> >>  >>
> >>  >>
> >>  >>
> >>  >>
> >>  >> On Nov 19, 2006, at 2:24 AM, Ani Anyanwu wrote:
> >>  >>
> >>  >>>  Prasanna
> >>  >>>
> >>  >>>  Well many would I suspect call it unbridled.
> >>  >>>
> >>  >>>  The following would generally receive aprotinin in my institution
> >>  >>>  1) reoperations
> >>  >>>  2) operations on the aortic arch or descending aorta
> >>  >>>  3) transplant and VAD procedures
> >>  >>>  4) operations on patients on clopidogrel
> >>  >>>  5) combined valvular and CABG
> >>  >>>  6) Patients with renal impairment
> >>  >>>  7) Patients where ability to tolerate transfusion or bleeding
> >>  >>> complications is thought to be marginal including - most
> >>  >>> patients  aged 70 or above, patients with severe lung disease,
> >>  >>> poor LV  function, severe pulmonary hypertension, multiple
> >>  >>> comorbidity etc.  Certainly almost all octogenrians would get
> >>  >>> aprotinin - even for CABG.
> >  > >>>  8) Paradoxically, young patients in their 20s or 30s (where
> >>  >>> avoidance of blood transfusion should be the goal in all patients)
> >>  >>>  9) Multiple valvular procedures (excluding tricuspid valve)
> >>  >>>  10) cases with anticipated bypass run more than 3 hours
> >>  >>> (including  complex mitral repairs)
> >>  >>>
> >>  >>>  As you can see there is not much left - so maybe it is
> >>  >>> unbridled!  As you implied we obviously would not use it for an
> >>  >>> ASD or isolated  AVR, but these constitute a small minority of
> >>  >>> our procedures.  Personally I would use it for practically every
> >>  >>> operation -  including all CABGs - but that is a personal opinion
> >>  >>> as I believe  there are non-hematological benefits of the drug
> >>  >>> and like you
> >>  >>  > strongly believe in blood conservation. I do not have any
> >>  >> interests
> >>  >>>  or links to industry.
> >>  >>>
> >>  >>>  Actually Ben brought up something that I had never thought of -
> >  > >>> correct me if I am wrong but Aprotinin is the only agent
> >>  >>> licensed  as a blood conservation agent for heart surgery?
> >>  >>>
> >>  >>>  Ani
> >>  >>>    ----- Original Message -----
> >>  >>>    From: psimha<mailto:prasannasimha at gmail.com>
> >>  >>>    To: OpenHeart-L at lists.hsforum.com<mailto:OpenHeart-
> >>  >>>  L at lists.hsforum.com>
> >>  >>>    Sent: Sunday, November 19, 2006 12:00 AM
> >>  >>>    Subject: Re: [HSF] Aprotinin
> >>  >>>
> >>  >>>
> >>  >>>    Ani - are you really using it "unbridled" or liberally ? Do
> >>  >>> you  use it
> >>  >>>    for an ASD or for a straight forward valve replacement ? or
> >>  >>> any  other
> >>  >>>    case with a short bypass run ?
> >>  >>>    I did not say I will not use it in a redo - in fact if you
> >>  >>> note my
> >>  >>>    original post I said I did use it in redo's ?
> >>  >>>    And Yes , I believe very strongly in blood conservation and
> >>  >>> believe that
> >>  >>>    Aprotinin is one (and not the only ) cog in the wheel.
> >>  >>  >   Prasanna
> >>  >>>
> >>  >>>    Ani Anyanwu wrote:
> >>  >>>>  Prasanna
> >>  >>>>
> >>  >>>>  We use aprotinin in an unbridled way and are certainly yet to
> >>  >>>> see  this price.
> >>  >>>>  - we have no more an incidence of renal failure than other
> >>  >>>> institutions have (this we know because incidence of dialysis
> >>  >>>> postop in all New York Hospitals is tracked by the State
> >>  >>>> Department of Health)
> >>  >>>>  - we have no suggestion of an increase in early vein graft
> >>  >>>> thrombosis (this should transform into higher periop MI and
> >>  >>>> mortality, our CABG mortality rate has remained around 1.5% last
> >>  >>>> 3  years)
> >>  >>>>  - we have not experienced any adverse events that caused us to
> >>  >>>> be  concerned about its use, except fatal thrombosis in 2
> >>  >>>> patients  with Factor V Lieden deficiency having circulatory
> >>  >>>> arrest so we  now routinely screen for this defect in all
> >>  >>>> circulatory arrest cases.
> >>  >>>>
> >>  >>>>  The price we are paying is a low incidence of transfusion of
> >>  >>>> blood  products and a low re-exploration rate (<2% last 2 years
> >>  >>>> even with  18% being redos and almost 20% aortic cases). Maybe
> >>  >>>> there are  other unknown adverse effects which will catch up
> >>  >>>> with us, but for  know they are unknown (and we wont be
> >>  >>>> responsible; remember it is  the drug companies not doctors
> >>  >>>> being sued for COX2 inhibitors).
> >>  >>>>
> >>  >>>>  Maybe when Mangano is bored he might do another study, and
> >>  >>>> then  what will you do? For those who use Amicar, how do we
> >>  >>>> really know  it is any safer - the drug is not even licensed for
> >>  >>>> human use in  many European countries. Perhaps even his next
> >>  >>>> study will be on  morbidity of plasma and platelet
> >>  >>>> transfusions....then what will we  do?
> >>  >>>>
> >>  >>>>  Ani
> >>  >>>>    ----- Original Message -----
> >>  >>>>    From:
> >>  >>>>
> prasannasimha<mailto:prasannasimha at gmail.com<mailto:prasannasimha at g
> >>  >>>> ma
> >>  >>>>  il.com>>
> >>  >>>>    To: OpenHeart-L at lists.hsforum.com<mailto:OpenHeart-
> >>  >>>>  L at lists.hsforum.com<mailto:OpenHeart-
> >>  >>>>  L at lists.hsforum.com<mailto:OpenHeart-L at lists.hsforum.com>>
> >>  >>>>    Sent: Saturday, November 18, 2006 9:37 PM
> >>  >>>>    Subject: Re: [HSF] Aprotinin
> >>  >>>>
> >>  >>>>
> >>  >>>>    The thing I want to say is that be it Vioxx / Aprotinin/blood/
> >  > >>>>  Oxygen -
> >>  >>>>    they are all drugs and have effects and side effects. The
> >>  >>>> present mess
> >>  >>>>    that the pharmacological companies are in is just because of
> >>  >>>> their
> >>  >>>>    unbridled enthusiasm (or greed) to ,make a quick buck and it
> >>  >>>> backfires
> >>  >>>>    on them. COX2 Inhibitors have a specific role unfortunately
> >>  >>>> I  even saw
> >>  >>>>    my dentist prescribing it for tooth pain !! Who marketed it
> >>  >>>> to  him as a
> >>  >>>>    good NSAID  ? I told him about the literature and my
> >>  >>>> concerns  (this was
> >>  >>>>    prior to Vioxx) . They were trying to market Valdecoxib for
> >>  >>>> post  cardiac
> >>  >>>>    surgery pain !!_ and I told them you should not be doing that
> >>  >>>> -  but did
> >>  >>>>    they listen ? and bang in a few months a controversy breaks
> >>  >>>> out.  The
> >>  >>>>    wife of colleague of mine was taking valdecoxib sample (she
> >  > >>>> is a  Doctor
> >>  >>>>    too) as the sample was around and the premenopausal lady
> >>  >>>> ended  up with a
> >>  >>>>    coronary thrombosis !!
> >>  >>>>    Every drug has a role and an indication based on good
> >>  >>>> clinical  judgment
> >>  >>  >>   - unfortunately we pay the price when its use is unbridled.
> >>  >>>>    Prasanna
> >>  >>>>
> >>  >>>>
> >>  hgrmd at aol.com<mailto:hgrmd at aol.com<mailto:hgrmd at aol.com<mailto:hgrm
> >>  >>>> d@
> >>  >>>>  aol.com>> wrote:
> >>  >>>>>  Prasanna and Ajit,
> >>  >>>>>    At the risk of great bodily harm from Ben, Ani, and others,
> >>  >>>>> I  again think the use of aprotinin should be limited as much
> >>  >>>>> as  possible.  I know there are cases where the benefit
> >>  >>>>> seemingly  outweighs the risk.  However, the mounting
> >>  >>>>> literature against it  is becoming increasingly compelling.  In
> >>  >>>>> addition, my own  impression, made years before any of this
> >>  >>>>> came out, was that the  drug increased the risk of ATN.  I'm
> >>  >>>>> also convinced that this has  the potential to be the Vioxx of
> >>  >>>>> cardiac surgery.  All I can say  is you guys who continue to
> >>  >>>>> indiscriminantly use it have got some  really big ones.
> >>  >>>>>  Hal
> >>  >>>>>
> >>  >>>>>
> >>  >>>>>  -----Original Message-----
> >>  >>>>>  From:
> >>  >>>>>
> prasannasimha at gmail.com<mailto:prasannasimha at gmail.com<mailto:pras
> >>  >>>>> an
> >>  >>>>>  nasimha at gmail.com<mailto:prasannasimha at gmail.com>>
> >>  >>>>>  To: OpenHeart-L at lists.hsforum.com<mailto:OpenHeart-
> >>  >>  >>> L at lists.hsforum.com<mailto:OpenHeart-
> >>  >>>>>  L at lists.hsforum.com<mailto:OpenHeart-L at lists.hsforum.com>>
> >>  >>>>>  Sent: Sat, 18 Nov 2006 1:00 PM
> >>  >>>>>  Subject: Re: [HSF] Aprotinin
> >>  >>>>>
> >>  >>>>>
> >>  >>>>>  Very Sorry used Aprotinin on my redo - can't help using it
> >>  >>>>> selectively !!
> >>  >>>>>  Prasanna
> >>  >>>>>
> >>  >>>>>  Ajit Damle wrote:
> >>  >>>>>
> >>  >>>>>>  Journal club critique >
> >>  >>>>>>  A disheartening story: Aprotinin in cardiac surgery >
> >>  >>>>>>  Lien M, Milbrandt E
> >>  >>>>>>
> >>  >>>>>>  Critical Care, 2006 10:317 ( 8 November 2006 )
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  Journal club critique
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  A disheartening story: Aprotinin in cardiac surgery
> >>  >>>>>>
> >>  >>>>>>  Marcus Lien1 and Eric B Milbrandt2 >
> >>  >>>>>>  1Clinical Fellow, Department of Critical Care Medicine,
> >>  >>>>>> University of
> >>  >>>>>>  Pittsburgh School of Medicine, Pittsburgh, Pennsylvania, USA
> >>  >>>>>>
> >>  >>>>>>  2Assistant Professor, Department of Critical Care Medicine,
> >>  >>>>>> University of
> >>  >>>>>>  Pittsburgh School of Medicine, Pittsburgh, Pennsylvania, USA
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  Critical Care 2006, 10:317 doi:10.1186/cc5072
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>>
> >>  >>>>>>>
> >>  >>>>>>  Evidence based medicine journal club critique edited by E B
> >>  >>>>>> Milbrant
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  The electronic version of this article is the complete one
> >>  >>>>>> and  can be found
> >>  >>>>>>  online at: http://ccforum.com/content/10/6/317<http://
> >>  >>>>>>  ccforum.com/content/10/6/317<http://ccforum.com/content/
> >>  >>>>>>  10/6/317<http://ccforum.com/content/10/6/317>>
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  Published 8 November 2006 >
> >>  >>>>>>
> >>  >>>>>>  C 2006 BioMed Central Ltd
> >>  >>>>>>
> >>  >>>>>>  Citation
> >>  >>>>>>
> >>  >>>>>>  Mangano DT, Tudor IC, Dietzel C: The risk associated with
> >  > >>>>>> aprotinin in
> >>  >>>>>>  cardiac surgery. N Engl J Med 2006, 354:353-365 [1].
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  Background
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  The majority of patients undergoing surgical treatment for ST-
> >>  >>>>>>  elevation
> >>  >>>>>>  myocardial infarction receive antifibrinolytic therapy to
> >>  >>>>>> limit  blood loss.
> >>  >>>>>>  This approach appears counterintuitive to the accepted
> >>  >>>>>> medical  treatment of
> >>  >>>>>>  the same condition - namely, fibrinolysis to limit
> >>  >>>>>> thrombosis.  Despite this
> >>  >>>>>>  concern, no independent, large-scale safety assessment has
> >>  >>>>>> been  undertaken.
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  Methods
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  Design and setting
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  Prospective observational cohort study in 69 institutions in
> >>  >>>>>> North and South
> >>  >>>>>>  America, the Middle East, Europe, and Asia.
> >>  >>>>>>
> >  > >>>>>>
> >>  >>>>>>  Subjects
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  4374 patients undergoing coronary-artery revascularization.
> >>  >>>>>> All  patients
> >>  >>>>>>  were >18 years old and completed a pre-surgery interview.
> >>  >>>>>> Patients were
> >>  >>>>>>  classified as undergoing primary surgery (no previous heart
> >>  >>>>>> surgery and no
> >>  >>>>>>  other surgery besides a coronary artery bypass graft), or
> >>  >>>>>> complex surgery
> >>  >>>>>>  (all other surgery).
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  Intervention
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  None.
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  Measurements
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  The authors prospectively assessed three agents (aprotinin
> >>  >>>>>> [1295  patients],
> >>  >>>>>>  aminocaproic acid [883], and tranexamic acid [822]) as
> >>  >>>>>> compared  with no
> >>  >>>>>>  agent (1374 patients) with regard to serious cardiovascular,
> >>  >>  >>>> renal, and
> >>  >>>>>>  cerebrovascular outcomes by propensity and multivariable
> >>  >>>>>> methods.
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  Results
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  In propensity-adjusted, multivariable logistic regression (C-
> >>  >>>>>>  index, 0.72),
> >>  >>>>>>  use of aprotinin was associated with a doubling in the risk
> >>  >>>>>> of  renal failure
> >>  >>>>>>  requiring dialysis among patients undergoing complex coronary-
> >>  >>>>>>  artery surgery
> >>  >>>>>>  (odds ratio, 2.59; 95 percent confidence interval, 1.36 to
> >>  >>>>>> 4.95)  or primary
> >>  >>>>>>  surgery (odds ratio, 2.34; 95 percent confidence interval,
> >>  >>>>>> 1.27  to 4.31).
> >>  >>>>>>  Similarly, use of aprotinin in the latter group was
> >>  >>>>>> associated  with a 55
> >>  >>>>>>  percent increase in the risk of myocardial infarction or
> >>  >>>>>> heart  failure (P <
> >>  >>>>>>  0.001) and a 181 percent increase in the risk of stroke or
> >>  >>>>>> encephalopathy (P
> >>  >>>>>>  = 0.001). Neither aminocaproic acid nor tranexamic acid was
> >>  >>>>>> associated with
> >>  >>>>>>  an increased risk of renal, cardiac, or cerebral events.
> >>  >>>>>> Adjustment
> >>  >>>>>>  according to propensity score for the use of any one of the
> >>  >>>>>> three agents as
> >>  >>>>>>  compared with no agent yielded nearly identical findings. All
> >>  >>  >>>> the agents
> >>  >>>>>>  reduced blood loss.
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  Conclusion
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  The association between aprotinin and serious end-organ
> >>  >>>>>> damage  indicates
> >>  >>>>>>  that continued use is not prudent. In contrast, the less
> >>  >>>>>> expensive generic
> >>  >>>>>>  medications aminocaproic acid and tranexamic acid are safe
> >>  >>>>>> alternatives.
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>>
> >>  >>>>>>  The medical and surgical approaches to acute ST-elevation
> >>  >>>>>> myocardial
> >>  >>>>>>  infarction present an interesting paradox. The medical
> >>  >>>>>> approach  focuses on
> >>  >>>>>>  fibrinolytic therapy. Due to concerns over bleeding, the
> >>  >>>>>> surgical approach
> >>  >>>>>>  avoids fibrinolytic agents and instead uses agents that
> >>  >>>>>> mitigate  bleeding,
> >>  >>>>>>  so called antifibrinolytic agents, which include aprotinin,
> >>  >>>>>> aminocaproic
> >>  >>>>>>  acid, and tranexamic acid. These agents were generally
> >>  >>>>>> considered safe based
> >>  >>>>>>  on a number of secondary analyses of studies that were not
> >>  >>>>>> primarily
> >>  >>>>>>  intended to assess safety. These relatively small studies
> >  > >>>>>> were  underpowered
> >>  >>>>>>  to detect adverse events and did not involve head-to-head
> >>  >>>>>> comparisons of the
> >>  >>>>>>  commonly used antifibrinolytic agents. Animal studies
> >>  >>>>>> suggest  that these
> >>  >>>>>>  agents have the potential to cause ischemic damage to
> >>  >>>>>> multiple  organ systems
> >>  >>>>>>  and small, largely single-center studies have suggested
> >>  >>>>>> increased graft
> >>  >>>>>>  thrombosis and renal dysfunction [2-6]. Ideally, the safety
> >>  >>>>>> of  these agents
> >>  >>>>>>  would be compared in a large, multi-center, randomized
> >>  >>>>>> controlled trial.
> >>  >>>>>>  However, because their use is embedded in practice and
> >>  >>>>>> because  regulatory
> >>  >>>>>>  approval of these agents differs by country, conducting such
> >>  >>>>>> a  trial will be
> >>  >>>>>>  difficult if not impossible.
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  To address the safety of these agents for cardiopulmonary
> >  > >>>>>> bypass  surgery,
> >>  >>>>>>  Mangano and colleagues [1] conducted a large, prospective,
> >>  >>>>>> observational
> >>  >>>>>>  cohort assessing aprotinin, aminocaproic acid, and
> >>  >>>>>> tranexamic  acid as
> >>  >>>>>>  compared to no agent in 4374 patients undergoing
> >>  >>>>>> revascularization. Because
> >>  >>>>>>  this was a prospective study, the authors were able to
> >>  >>>>>> collect a  wealth of
> >>  >>>>>>  clinical information, including approximately 7500 data
> >>  >>>>>> fields  per patient.
> >>  >>>>>>  This permitted consideration of variables that might
> >>  >>>>>> influence  both choice
> >>  >>>>>>  of antifibrinolytic agent and clinical outcome. The authors
> >>  >>>>>> used a
> >>  >>>>>>  propensity score based on 45 treatment-selection covariates
and
> >>  >>>>>>  multivariable modeling to control for baseline differences
> >>  >>>>>> between groups.
> >>  >>>>>>  In doing so, they found that aprotinin, but not aminocaproic
> >>  >>>>>> acid or
> >>  >>>>>>  tranexamic acid, was associated with serious cardiovascular,
> >>  >>>>>> renal, and
> >>  >>>>>>  cerebrovascular adverse events. Furthermore, a dose-response
> >>  >>>>>> relationship
> >>  >>>>>>  was demonstrated, strengthening the inference of causality.
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  The main weakness of this study is that the authors failed to
> >>  >>  >>>> report details
> >>  >>>>>>  of the surgery itself, such as whether the surgery was on
> >>  >>>>>> vs.  off-pump, time
> >>  >>>>>>  on pump, and number of vessels bypassed. These variables are
> >>  >>>>>> likely to
> >>  >>>>>>  influence not only choice of antifibrinolytic agent but also
> >>  >>>>>> outcome, and
> >>  >>>>>>  are, therefore, a source of indication bias that could
> >>  >>>>>> reflect  unfavorably
> >>  >>>>>>  on aprotinin.
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  Based on the results of this study and those of another
> >>  >>>>>> observational study
> >>  >>>>>>  suggesting renal toxicity [7], the United States Food and Drug
> >>  >>>>>>  Administration (FDA) held an advisory committee meeting
> >>  >>>>>> September 21, 2006
> >>  >>>>>>  to consider the cardiovascular safety of aprotinin. Because
> >>  >>>>>> of  concerns
> >>  >>>>>>  about the methodology of the study by Mangano and colleagues
> >>  >>>>>> and  because it
> >>  >>>>>>  was the only study to suggest cardiovascular adverse events
> >>  >>>>>> [8],  the
> >>  >>>>>>  advisory committee concluded that there was insufficient
> >>  >>>>>> evidence to support
> >>  >>>>>>  changing the cardiovascular safety labeling of the drug.
> >>  >>>>>> However, just six
> >>  >>>>>>  days after the committee met, it was revealed that the
> >>  >>>>>> drug's  manufacturer,
> >>  >>  >>>> Bayer, had preliminary results from an observational study of
> >>  >>>>>>  67,000 cardiac
> >>  >>>>>>  bypass patients that suggested aprotinin was associated with
> >>  >>>>>> increased risk
> >>  >>>>>>  of death, renal dysfunction, congestive heart failure, and
> >>  >>>>>> stroke [9]. The
> >>  >>>>>>  FDA subsequently issued a statement indicating it was unaware
> >>  >>>>>> of  this study
> >>  >>>>>>  when the advisory committee met and that it is evaluating
> >>  >>>>>> the  results of
> >>  >>>>>>  this study and the potential implications for the use of
> >>  >>>>>> aprotinin [10]. In
> >>  >>>>>>  the mean time, the FDA suggests that physicians who use
> >>  >>>>>> aprotinin should
> >  > >>>>>>  carefully monitor patients for the occurrence of toxicity,
> >>  >>>>>> particularly to
> >>  >>>>>>  the kidneys, heart, or brain, and promptly report observed
> >>  >>>>>> adverse events.
> >>  >>>>>>  They go on to recommend that physicians should consider
> >>  >>>>>> limiting  aprotinin
> >>  >>>>>>  use to those situations where the clinical benefit of
> >>  >>>>>> reduced  blood loss is
> >>  >>>>>>  essential to medical management of the patient and outweighs
> >>  >>>>>> the  potential
> >>  >>>>>>  risks.
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  Recommendation >
> >>  >>>>>>
> >>  >>>>>>  The weight of evidence suggests that aprotinin increases the
> >>  >>>>>> risk for a poor
> >>  >>>>>>  outcome among patients undergoing cardiac operations. Not
> >>  >>>>>> only  is this drug
> >>  >>>>>>  very expensive, it seems to be toxic. Although the risk of
> >>  >>>>>> excessive
> >>  >>>>>>  bleeding is certainly a cause for concern in certain
> >>  >>>>>> patients,  and treatment
> >  > >>>>>>  with aprotinin can decrease blood loss in selected patients,
> >>  >>>>>> data are
> >>  >>>>>>  lacking to show that administration of this agent actually
> >>  >>>>>> improves
> >>  >>>>>>  survival.
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  Competing interests
> >>  >>>>>>
> >>  >>>>>>  The authors declare that they have no competing interests.
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>>
> >>  >>>>>>  1. Mangano DT, Tudor IC, Dietzel C: The risk associated with
> >>  >>>>>> aprotinin in
> >>  >>>>>>  cardiac surgery.
> >>  >>>>>>
> >>  >>>>>>  N Engl J Med 2006, 354:353-365. >
> >>  >>>>>>
> >>  >>>>>>  2. Cosgrove DM III, Heric B, Lytle BW, Taylor PC, Novoa R,
> >>  >>>>>> Golding LA,
> >>  >>>>>>  Stewart RW, McCarthy PM, Loop FD: Aprotinin therapy for
> >>  >>>>>> reoperative
> >>  >>>>>>  myocardial revascularization: a placebo-controlled study.
> >>  >>>>>>
> >>  >>>>>>  Ann Thorac Surg 1992, 54:1031-1036.
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  3. D'Ambra MN, Akins CW, Blackstone EH, Bonney SL, Cohn LH,
> >>  >>>>>> Cosgrove DM,
> >>  >>>>>>  Levy JH, Lynch KE, Maddi R: Aprotinin in primary valve
> >>  >>>>>> replacement and
> >>  >>>>>>  reconstruction: a multicenter, double-blind, placebo-
> >>  >>>>>> controlled  trial.
> >>  >>>>>>
> >>  >>>>>>  J Thorac Cardiovasc Surg 1996, 112:1081-1089
> >>  >>>>>>
> >>  >>>>>>
> >>  >>>>>>  4. Feindt PR, Walcher S, Volkmer I, Keller HE, Straub U,
> >>  >>>>>> Huwer  H, Seyfert
> >>  >>>>>>  UT, Petzold T, Gams E: Effects of high-dose aprotinin on
> >>  >>>>>> renal  function in
> >>  >>>>>>  aortocoronary bypass grafting.
> >>  >>>>>>
> >>  >>>>>>  Ann Thorac Surg 1995, 60:1076-1080 >
> >>  >>>>>>
> >>  >>>>>>  5. Sundt TM III, Kouchoukos NT, Saffitz JE, Murphy SF,
> >>  >>>>>> Wareing  TH, Stahl
> >>  >>>>>>  DJ: Renal dysfunction and intravascular coagulation with
> >>  >>>>>> aprotinin and
> >>  >>>>>>  hypothermic circulatory arrest.
> >>  >>  >>>>
> >>  >>>>>>  Ann Thorac Surg 1993, 55:1418-1424 >
> >>  >>>>>>
> >>  >>>>>>  6. Umbrain V, Christiaens F, Camu F: Intraoperative coronary
> >>  >>>>>> thrombosis:
> >>  >>>>>>  can aprotinin and protamine be incriminated?
> >>  >>>>>>
> >>  >>>>>>  J Cardiothorac Vasc Anesth 1994, 8:198-201 >
> >>  >>>>>>
> >>  >>>>>>  7. Karkouti K, Beattie WS, Dattilo KM, McCluskey SA, Ghannam
> >>  >>>>>> M,  Hamdy A,
> >>  >>>>>>  Wijeysundera DN, Fedorko L, Yau TM: A propensity score case-
> >>  >>>>>> control
> >>  >>>>>>  comparison of aprotinin and tranexamic acid in
high-transfusion-
> >>  >>>>>>  risk cardiac
> >>  >>>>>>  surgery.
> >>  >>>>>>
> >>  >>>>>>  Transfusion 2006, 46:327-338 >
> >>  >>>>>>
> >>  >>>>>>  8. Hughes S: Aprotinin safety again in spotlight as new
> >>  >>>>>> study  suggests
> >>  >>>>>>  increased cardiac events.
> >>  >>>>>>
> >>  >>>>>>  http://www.medscape.com/viewarticle/545400<http://
> >>  >>>>>>  www.medscape.com/viewarticle/545400<http://www.medscape.com/
> >>  >>>>>>  viewarticle/545400<http://www.medscape.com/viewarticle/
> >>  >>>>>> 545400>> >
> >>  >>>>>>  October 2, 2006 >
> >>  >>>>>>  9. Harris G: FDA says Bayer failed to reveal drug risk study.
> >>  >>>>>>
> >>  >>>>>>  [http://www.nytimes.com/2006/09/30/health/30fda.html] New
> >>  >>>>>> York  Times >
> >>  >>>>>>
> >>  >>>>>>  10. US Food and Drug Administration: FDA Public Health
> >>  >>>>>> Advisory:  Aprotinin
> >>  >>>>>>  Injection (marketed as Trasylol).
> >>  >>>>>>
> >>  >>>>>>  [http://www.fda.gov/cder/drug/advisory/aprotinin20060929.htm]
>
> >>  >>  >>>> September 29, 2006 >
> >  > >>>>>>
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> >>
> __________________________________________________________________
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> >>  >> -----------------------------------------
> >>  >>
> >>  >> _______________________________________________
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> >>  >> -----------------------------------------
> >>  >
> >>  >
> >>  > --
> >>  > Ben Bidstrup FRACS FRCSEd FEBCTS
> >>  > Consultant Cardiothoracic Surgeon
> >>  > _______________________________________________
> >>  > OpenHeart-L mailing list
> >>  >
> >>  > Send postings to:
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> >>  > -----------------------------------------
> >>
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> >>
> >>  All messages transmitted by the OpenHeart-L are subject to the
policies
> >and
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> >>  -----------------------------------------
> >
> >_______________________________________________
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and
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> >-----------------------------------------
> 
> 
> --
> Ben Bidstrup FRACS FRCSEd FEBCTS
> Consultant Cardiothoracic Surgeon
> _______________________________________________
> OpenHeart-L mailing list
> 
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> All messages transmitted by the OpenHeart-L are subject to the policies
and
> disclaimers posted at:
> http://www.hsforum.com/listdisclaim
> -----------------------------------------



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